ADVERTISEMENT RETURN TO ISSUELetterNEXTPhysicochemical High Throughput Screening: Parallel Artificial Membrane Permeation Assay in the Description of Passive Absorption Processe...
Abstract This review describes simple and useful concepts for predicting and tuning the p K a values of basic amine centers, a crucial step in the optimization of physical and A...
Abstract In a systematic fluorine scan of a rigid inhibitor to map the fluorophilicity/fluorophobicity of the active site in thrombin, one or more F substituents were introduced...
Abstract A series of 16 tricyclic thrombin inhibitors was prepared by using the 1,3‐dipolar cycloaddition of azomethine ylides derived from 3‐ or 4‐hydroxyproline and 4‐bromoben...
h-index: Number of publications with at least h citations each.